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Frontiers in New Drug Discovery: From Molecular Targets to Preclinical Trials

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Streptococci; antimicrobials; QSAR; MD simulation; Kunitz-type peptides; neuroprotective activity; sea anemones; TRPV1; P2X7R; Parkinson’s disease (PD); diffuse large B cell lymphoma (DLBCL); deep neural network; drug discovery; drug combination; biomarker; cancer severity; cancer prognosis; MAFB; tumor-associated macrophages; prostate cancer; photodynamic therapy; magnetic resonance imaging; ex vivo; anti-inflammatory substance; N-acylhydrazone; naphthyl-N-acylhydrazone; LASSBio-1524 analogues; phosphacoumarin; azomethine ylide; cycloaddition; anti-cancer; cytotoxicity; quantum chemistry; pravastatin; metformin; radiation-induced intestinal injury; minipigs; epithelial regeneration; inflammation; arylazo sulfones; DNA binding; DNA cleavage; DNA photocleavage; A375 melanoma cells; molecular docking; radicals; N–S bond homolysis; platinum(II); five-coordinate complexes; glycoconjugation; cytotoxic activity; protein X-ray structure; lipophilicity; natural products; acetylcholinesterase inhibitors; butyrylcholinesterase inhibitors; Alzheimer’s disease; central nervous system; n/a

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